Color: | White | Order: | Characteristic |
---|---|---|---|
Assay: | NLT 99% | Other Name: | 3-Amino-4-phenylbutyric Acid Hydrochloride |
MOQ: | 100G | Cas No.: | 148553-50-8 |
Apprarence: | Crystal Powder | Usage: | Relieve Pain |
High Light: | Pregabalin Pain Relief Powder,Anticonvulsant Pain Relief Powder,CAS 148553-50-8 |
Pregabalin Pain Relief Powder CAS 148553-50-8 For Anticonvulsant
1. Production Information Of Pregabalin
Pregabalin, chemical name (s) - 3-aminomethyl-5-methylcaproic acid, molecular formula c8h17no2, is an antiepileptic drug, which is mainly used to treat postherpetic neuralgia clinically.Pregabalin is an analogue of γ-aminobutyric acid (GABA), similar in structure and function to gabapentin, and has antiepileptic, analgesic and anxiolytic activities. The antiepileptic mechanism of pregabalin is still unclear. In laboratory studies, pregabalin has anticonvulsant activity on various epilepsy models; After oral administration, pregabalin takes effect within 30 minutes for acute toothache, lasting about 5 hours, and takes effect within 1 week for diabetic neuropathy. The peak time was about 1 h and the bioavailability was 90%. It is less metabolized in liver, 92% ~ 99% excreted by kidney in original form, less than 0.1% excreted by faeces in oral dose, with half-life of 5-6.5h
Product Name: | Pregabalin |
MW | 159.22600 |
CAS Number | 148553-50-8 |
PSA |
63.32000
|
Purity | 99% |
Storage | stay in dry, cool and well-sealed |
Package | 1kg plastic drum |
Appearance | White powder |
Application |
Relieve pain |
Less on drying |
NMT 1.0% |
Melting point | 194-196ºC |
Heavy metals | 10 ug/gMax |
Loss On Drying | ≤0.5% |
2. Funcation Of Pregabalin
1. Neuropathic pain and postherpetic neuralgia in diabetic peripheral neuropathy.
2. Adjuvant treatment of partial seizures.
3. It can also be used for anxiety disorder, social phobia and arthritis
4. Pregabalin can enhance the sedative effect of central nervous system inhibitors.
5. Pregabalin can enhance the sedative effect of alcohol.
6. Food can reduce the bioavailability of pregabalin