Color: | White | Order: | Characteristic |
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Assay: | NLT99% | Other Name: | 3-Amino-4-phenylbutyric Acid Hydrochloride |
MOQ: | 10G | Cas No.: | 3060-41-1 |
Apprarence: | Crystal Powder | Usage: | Nootropics |
High Light: | Nootropics Phenibut Powder,GABA Phenibut Powder,CAS 1078-21-3 |
99% Phenibut HCL / Fenibut HCL Nootropics Powder
1. Production Information Of Phenibut
Also known as "4-Amino-3-Phenylbutyric Acid," Phenibut is a non-prescription pharmaceutical that is actually a GABA molecule with the addition of a phenyl group. Russian researchers discovered that by changing GABA into 4-Amino-3-Phenylbutyric Acid, it was able to cross more easily into the nervous system & across the blood-brain barrier. Since it is a GABA, an inhibitory neurotransmitter, derivative, Phenibut increases GABA levels.
Product Name: | Phenibut / Fenibut | |
MW | 215.68 | |
CAS Number | 3060-41-1 | |
EINECS: |
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Purity | 99% | |
Storage | stay in dry, cool and well-sealed | |
Package | 25kgs plastic drum | |
Appearance | White powder | |
Application |
Nootropics |
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Less on drying |
NMT 1.0% |
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Melting point | 194 ~ 202ºC | |
Heavy metals | 10 ug/gMax | |
Loss On Drying | ≤0.5% |
2. Funcation Of Phenibut
Phenibut is a central depressant and analog of the inhibitory neurotransmitter γ-aminobutyric acid (GABA), or a GABA analogue. The addition of a phenyl ring allows phenibut to cross the blood-brain barrier. Phenibut was developed in the Soviet Union in the 1960s, and has since been used there as a pharmaceutical drug to treat a wide range of ailments, including posttraumatic stress disorder, anxiety, depression, asthenia, insomnia, alcoholism, stuttering, and vestibular disorders, and other conditions.
Phenibut is a close structural analogue of GABA, as well as of baclofen (β-(4-chlorophenyl)-GABA) and GABOB (β-hydroxy-GABA). Phenibut is believed to act as a selective GABAB receptor agonist; studies are conflicting as to whether phenibut also acts as a GABAA receptor agonist. More recently, phenibut has been found to act preferentially as a blocker of α2δ subunit-containing voltage-gated calcium channels, similarly to gabapentin. As such, by definition, phenibut is a gabapentinoid.